2021年度分子創薬化学セミナー（後期） - 徳島大学薬学部?大学院

第410回 (2021. 12. 22)
担当者:中尾允泰
文献名:"Zinc-Catalyzed β-Functionalization of Cyclopropanols via Enolized Homoenolate"
Y. Sekiguchi and N. Yoshikai
J. Am. Chem. Soc., 143 (44), 18400-18405 (2021).

第409回 (2021. 12. 18)
担当者:竹原未来子
文献名:"Enantioselective Rh(II)-Catalyzed Desymmetric Cycloisomerization of Diynes: Constructing Furan-Fused Dihydropiperidines with an Alkyne-Substituted Aza-Quaternary Stereocenter"
R. Wu, J. Lu, T. Cao, J. Ma, K. Chen, and S. Zhu
J. Am. Chem. Soc., 143 (36), 14916-14925 (2021).

第408回 (2021. 12. 18)
担当者:岡本麻里衣
文献名:"Total Synthesis of (+)-Cyclobutastellettolide B"
Z. Zhang, S. Chen, F. Tang, K. Guo, X. -T. Liang, J. Huang, and Z. Yang
J. Am. Chem. Soc., 143 (43), 18287-18293 (2021).

第407回 (2021. 12. 11)
担当者:山口真生
文献名:"Siloxy Esters as Traceless Activators of Carboxylic Acids: Boron-Catalyzed Chemoselective Asymmetric Aldol Reaction"
T. Fujita, M. Yamane, W. M. C. Sameera, H. Mitsunuma, and M. Kanai
Angew. Chem. Int. Ed., 60 (46), 24598-24604 (2021).

第406回 (2021. 12. 11)
担当者:藤井千恵子
文献名:"Ynamides as Three-Atom Components in Cycloadditions: An Unexplored Chemical Reaction Space"
D. Campeau, A. Pommainville, and F. Gagosz
J. Am. Chem. Soc., 143 (25), 9601-9611 (2021).

第405回 (2021. 12. 4)
担当者:舟田遥乃
文献名:"Enantioconvergent Cu-Catalyzed Radical C–N Coupling of Racemic Secondary Alkyl Halides to Access α-Chiral Primary Amines"
Y. -F. Zhang, X. -Y. Dong, J. -T. Cheng, N. -Y. Yang, L. -L. Wang, F. -L. Wang, C. Luan, J. Liu, Z. -L. Li, Q. -S. Gu, and X. -Y. Liu
J. Am. Chem. Soc., 143 (37), 15413-15419 (2021).

第404回 (2021. 12. 4)
担当者:久保明音
文献名:"Aryl Amination Using Soluble Weak Base Enabled by a Water-Assisted Mechanism"
S. H. Lau, P. Yu, L. Chen, C. B. Madsen-Duggan, M. J. Williams, and B. P. Carrow
J. Am. Chem. Soc., 142 (47), 20030-20039 (2020).

第403回 (2021. 11. 20)
担当者:堀越拳
文献名:"Total Synthesis of (–)-Strempeliopine"
X. Zeng and D. L. Boger
J. Am. Chem. Soc., 143 (31), 12412-12417 (2021).

第402回 (2021. 11. 6)
担当者:僧津真之介
文献名:"Catalytic Asymmetric Aza-Diels–Alder Reaction of Ketimines and Unactivated Dienes"
Q. Zhao, Y. Li, Q. -X. Zhang, J. -P. Cheng, and X. Li
Angew. Chem. Int. Ed., 60 (32), 17608-17614 (2021).

第401回 (2021. 11. 6)
担当者:今橋縁
文献名:"Enantioselective and Diastereodivergent Synthesis of Spiroindolenines via Chiral Phosphoric Acid-Catalyzed Cycloaddition"
T. Varlet, M. Matisic, E. V. Elslande, L. Neuville, and V. Gandon
J. Am. Chem. Soc., 143 (30), 11611-11619 (2021).

第400回 (2021. 10. 30)
担当者:田原昌和
文献名:"Catalytic Asymmetric Cyanoalkylation of Electron-Deficient Olefins with Potassium Cyanide and Alkyl Halides"
K. Ohmatsu, Y. Morita, M. Kiyokawa, and T. Ooi
J. Am. Chem. Soc., 143 (29), 11218-11224 (2021).

第399回 (2021. 10. 30)
担当者:岡崎遼太郎
文献名:"Direct Access to α-Aminosilanes Enabled by Visible-Light-Mediated Multicomponent Radical Cross-Coupling"
X. Yu, C. G. Daniliuc, F. A. Alasmary, and A. Studer
Angew. Chem. Int. Ed., 60 (43), 23335-23341 (2021).

その他の分子創薬化学セミナー * Molecular Medicinal Chemistry Seminar