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80.
Development of Ribityllumazine Analogue as Mucosal-Associated Invariant T Cell Ligands
Takasaki, R.; Ito, E.; Nagae, M.; Takahashi, Y.; Matsuoka, T.; Yasue, W.; Arichi, N.; Ohno, H.*; Yamasaki, S.*; Inuki, S.*
J. Am. Chem. Soc. 2024, 146, 29964–29976.
doi: org/10.1021/jacs.4c12997



79.
Approach to Spirocyclohexadienes via Visible Light-Mediated ipso-Cyclization of Amino Acid Derivatives with N-(2-Phenyl)benzoyl Groups
Yoshida, Y.; Takeuchi, H.; Arichi, N.; Oishi, S.; Ohno, H.*; Inuki, S.*
Asian J. Org. Chem. 2024, 13, e202400140.
doi: org/10.1002/ajoc.202400140

78.
Structure-Activity Relationship Studies of Tetrahydroquinolone Derivatives as GPR41 Modulators
Inuki, S.; Miyamoto, J.; Hashimoto, N.; Shimizu, H.; Tabuchi, H.; Kawai, A.; Greiner, L. C.; Kimura, I.*; Ohno, H.*
Bioorg. Med. Chem. Lett. 2024, 107, 129758.
doi: org/10.1016/j.bmcl.2024.129758

77.
Synthesis of Labionin and Avionin Precursors via Nitrogen-Centred-Radical-Triggered 1,5-HAT Reaction of Tris Derivatives
Yamaguchi, A.; Obiya, N.; Arichi, N.; Oishi, S.; Ohno, H.*; Inuki, S.*
Org. Biomol. Chem. 2024, 22, 2049–2055.
doi: org/10.1039/D3OB02037A

76.
Synthesis of Sulfilimines via Visible-Light-Mediated Triplet Energy Transfer to Sulfonyl Azides
Arichi, N.*; Amano, T.; Wu, S.; Inuki, S.; Ohno, H.*
Chem. Eur. J. 2024, 30, e202401842.

75.
Chemical Synthesis of Interleukin?6 for Mirror-Image Screening
Aoki, K.; Maeda, K.; Inuki, S.; Ohno, H.; Nonaka, M.*; Oishi, S.*
Bioconjug. Chem. 2024, 35, 1190–1199..

74.
Mirror-Image Human Serum Albumin Domain III as a Tool for Analyzing Site II-Dependent Molecular Recognition
Iwamoto, N.; Kai, T.; Inuki, S.; Ohno, H.; Maeda, H.; Watanabe, H.; Maruyama, T.; Oishi, S.*
Bioconjug. Chem. 2024, 35, 816–825.

73.
Construction of the Akuammiline Alkaloid Core Structure via Stereoselective E-Ring Formation
Hashimoto, N.; Taguchi, J.; Kasagi, T.; Arichi, N.; Inuki, S.; Ohno, H.*
J. Org. Chem. 2024, 89, 10388–10392.

72.
Engineering a Low-Immunogenic Mirror-Image VHH against Vascular Endothelial Growth Factor
Aoki, K.; Higashi, K.; Oda, S.; Manabe, A.; Maeda, K.; Morise, J.; Oka, S.; Inuki, S.; Ohno, H.; Oishi, S.*; Nonaka, M.*
ACS Chem. Biol. 2024, 19, 1194–1205.

71.
Synthetic Study of Full-length Hepatitis B Virus Core Protein and Its Capsid Formation
Aoki, K.; Tsuda, S.; Ogata, N.; Kataoka, M.; Sasaki, J.; Inuki, S.; Ohno, H.; Watashi, K.; Yoshiya, T.; Oishi, S.*
Org. Biomol. Chem. 2024, 22, 2218–2225.

70.
Synthetic Studies on the Extracellular Domain of the T Cell Immunoreceptor with Immunoglobulin and Immunoreceptor Tyrosine-Based Inhibitory Motif Domain (TIGIT) Using Trt-K10 Solubilizing Tags
Iwamoto, N.; Sakaki, J.; Ohno, S.; Aoki, K.; Usui, Y.; Inuki, S.; Ohno, H.; Oishi, S.*
Bioorg. Med. Chem. 2024, 99, 117585.

69.
Sulfated Bile Acid is a Host-derived Ligand for MAIT Cells
Ito, E.; Inuki, S.; Izumi, Y.; Takahashi, M.; Dambayashi, Y.; Ciacchi, L.; Awad, W.; Takeyama, A.; Shibata, K.; Mori, S.; Mak, J. Y. W.; Fairlie, D. P.; Bamba, T.; Ishikawa, E.; Nagae, M.; Rossjohn, J.; Yamasaki, S.*
Sci. Immunol. 2024, 9, eade6924.

68.
Gold(I)-Catalyzed Cascade Cyclization of Alkynyl Indoles for the Stereoselective Construction of the Quaternary Carbon Center of Akuammiline Alkaloids
Hashimoto, N.; Taguchi, J.; Arichi, N.; Inuki, S.; Ohno, H.*
J. Org. Chem. 2023, 88, 17306–17321.

67.
Establishment of an MR1-Presentation Reporter Screening System and Identification of Phenylpropanoid Derivatives as MR1 Ligands
Matsuoka, T.; Hattori, A.; Oishi, S.; Araki, M.; Ma, B.; Fujii, T.; Arichi, N.; Okuno, Y.; Kakeya, H.; Yamasaki, S.; Ohno, H.*; Inuki, S.*
J. Med. Chem. 2023, 66, 12520–12535.
doi: org/10.1021/acs.jmedchem.3c01122

66.
Archaeal Glycerolipids Are Recognized by C-type Lectin Receptor Mincle
Oka, S.; Watanabe, M.; Ito, E.; Takeyama, A.; Matsuoka, T.; Takahashi, M.; Izumi, Y.; Arichi, N.; Ohno, H.*; Yamasaki, S.*; Inuki, S.*
J. Am. Chem. Soc. 2023, 145, 18538–18548.
doi: org/10.1021/jacs.3c05473

65.
Construction of a Bicyclo[2.2.2]octene Skeleton via a Visible-Light-Mediated Radical Cascade Reaction of Amino Acid Derivatives with N-(2-Phenyl)benzoyl Groups
Yoshida, Y.; Takeuchi, H.; Nakagawa, K.; Fujii, T.; Arichi, N.; Oishi, S.; Ohno, H.*; Inuki, S.*
Org. Lett. 2023, 25, 4846–4851.
doi: org/10.1021/acs.orglett.3c01586

64.
Variational Autoencoder-Based Chemical Latent Space for Large Molecular Structures with 3D Complexity
Ochiai, T.; Inukai, T.; Akiyama, M.; Furui, K.; Ohue, M.; Matsumori, N.; Inuki, S.; Uesugi, M.; Sunazuka, T.; Kikuchi, K.; Kakeya, H.; Sakakibara, Y.*
Commun. Chem. 2023, https://doi.org/10.1038/s42004-023-01054-6.

63.
Mirror-Image Single-Domain Antibody for a Novel Non-immunogenic Drug Scaffold
Aoki, K.; Manabe, A.; Kimura, H.; Katoh, Y.; Inuki, S.; Ohno, H.; Nonaka, M.; Oishi, S.*
Bioconjug. Chem. 2023, 34, 2055–2065.

62.
Design and Synthesis of Monobody Variants with Low Immunogenicity
Iwamoto, N.; Sato, Y.; Manabe, A.; Inuki, S.; Ohno, H.; Nonaka, M.; Oishi, S.*
ACS Med. Chem. Lett. 2023, 14, 1596–1601.

61.
Design of Synthetic Surrogates for the Macrolactone Linker Motif in Coibamide A
Suzuki, R.; Mattos, D. R.; Kitamura, T.; Tsujioka, R.; Kobayashi, K.; Inuki, S.; Ohno, H.; Ishmael, J. E.; McPhail, K. L.; Oishi, S.*
ACS Med. Chem. Lett. 2023, 14, 1344–1350.

60.
Gold(I)�\Catalyzed Bis�\Cyclization of Allenynes for the Synthesis of Strained and Planar Polycyclic Compounds
Tsuno, H.; Shen, J.; Komatsu, H.; Arichi, N.; Inuki, S.; Ohno, H.*
Angew. Chem., Int. Ed. 2023, 62, e202307532.

59.
Alkoxymigration onto α-Imino Gold Carbenes for Constructing Propellane-Type Indolines
Greiner, L. C.; Arichi, N.; Inuki, S.; Ohno, H.*
Asian J. Org. Chem. 2023, 12, e202300232.

58.
Discovery of Bis-sulfonamides as Novel Inhibitors of Mitochondrial NADH-Quinone Oxidoreductase (Complex I)
Tsuji, A.; Masuya, T.; Arichi, N.; Inuki, S.; Murai, M.; Miyoshi, H.; Ohno, H.*
ACS Med. Chem. Lett. 2023, 13, 211–216.

57.
Gold(I)-Catalyzed Benzylic C(sp3)H Functionalizations: Divergent Synthesis of Indole[a]- and [b]-Fused Polycycles
Greiner, L. C.; Arichi, N.; Inuki, S.; Ohno, H.*
Angew. Chem., Int. Ed. 2023, 62, e202213653.

56.
Host Metabolic Benefits of Prebiotic Exopolysaccharides Produced by Leuconostoc mesenteroides
Miyamoto, J; Shimizu, H.; Hisa, K.; Matsuzaki, C.; Inuki, S.; Ando, Y.; Nishida, A.; Izumi, A.; Yamano, M.; Ushiroda, C.; Irie, J.; Katayama, T.; Ohno, H.; Itoh, H.; Yamamoto, K.; Kimura, I.*
Gut Microbes 2023, 15, 2161271.

55.
The Identification of Novel Small Extracellular Vesicle (sEV) Production Modulators Using Luciferase�\Based sEV Quantification Method
Yamamoto, A.; Takahashi, Y.*; Inuki, S.; Nakagawa, S.; Nakao, K.; Ohno, H.; Doi, M.; Takakura, Y.
J. Extracell. Biol. 2022, 1, e62.

54.
A Methylbenzimidazole Derivative Regulates Mammalian Circadian Rhythms by Targeting Cryptochrome Proteins
Yagi, M.; Miller, S.; Nagai, Y.; Inuki, S.; Sato, A.; Hirota, T.*
F1000Research 2022, 11, 1016.

53.
Chemical Synthesis and Evaluation of Exopolysaccharide Fragments Produced by Leuconostoc mesenteroides strain NTM048
Inuki, S.*; Tabuchi, H.; Matsuzaki, C.; Yonejima, Y.; Hisa, K.; Kimura, I.; Yamamoto, K.; Ohno, H.*
Chem. Pharm. Bull. 2022, 70, 155–161.
doi: org/10.1248/cpb.c21-00919

52.
Design of Coibamide A Mimetics with a Simplified Macrocyclic Scaffold: An SAR Study to Improve the Cellular Bioactivity
Kitamura, T.; Suzuki, R.; Inuki, S.; Ohno, H.; McPhail, K. L.; Oishi, S.*
ACS Med. Chem. Lett. 2022, 13, 105–110.

51.
Construction of Tricyclic Nitrogen Heterocycles by Gold(I)-Catalyzed Cascade Cyclization of Allenynes and Its Application to Polycyclic π-Electron Systems
Komatsu, H.; Ikeuchi, T.; Tsuno, H.; Arichi, N.; Yasui, K.; Oishi, S.; Inuki, S.; Fukazawa, A.*; Ohno, H.*
Angew. Chem., Int. Ed. 2021, 60, 27019–27025.

50.
Access to Benzannulated Indole-Fused Medium-Sized Rings through Gold(I)-Catalyzed Cascade Cyclization of Azido-alkynes
Greiner, L. C.; Inuki, S.; Arichi, N.; Oishi, S.; Suzuki, R.; Iwai, T.; Sawamura, M.; Hashmi, A. S. K.; Ohno, H.*
Chem. Eur. J. 2021, 27, 12992–12997.

49.
The Effects of 5�\OP�\RU Stereochemistry on Its Stability and MAIT�\MR1 Axis
Matsuoka, T.; Motozono, C.; Hattori, A.; Kakeya, H.; Yamasaki, S.; Oishi, S.; Ohno, H.*; Inuki, S.*
ChemBioChem 2021, 22, 672–678.
doi: org/10.1002/cbic.202000466

48.
Identification of a Novel Indoleamine 2,3-Dioxygenase Inhibitor Bearing an Eight-Membered Ring Fused Indole Scaffold and its Structure Activity Relationship
Yamaguchi, A.; Inuki, S.*; Ohta, K.; Oishi, S.; Asai, A.; Ohno, H.*
Heterocycles 2021, 103, 331–347.

47.
Total Synthesis of Zephycarinatines via Photocatalytic Reductive Radical ipso-Cyclization
Takeuchi, H.; Inuki, S.*; Nakagawa, K.; Kawabe, T.; Ichimura, A.; Oishi, S.; Ohno, H.*
Angew. Chem., Int. Ed. 2020, 59, 21210–21215.
doi: org/10.1002/anie.202009399

46.
Polar Functional Group-Containing Glycolipid CD1d Ligands Modulate Cytokine-Biasing Responses and Prevent Experimental Colitis
Inuki, S.; Hirata, N.; Kashiwabara, E.; Kishi, J.; Aiba, T.; Teratani, T.; Nakamura, W.; Kojima, Y.; Maruyama, T.; Kanai, T.; Fujimoto, Y.*
Sci. Rep. 2020, 10, 15766.
doi: 10.1038/s41598-020-72280-4

45.
Total Synthesis of (+)-Polyoxamic Acid via Visible-Light-Mediated Photocatalytic β-Scission and 1,5-Hydrogen Atom Transfer of Glucose Derivative
Matsuoka, T.; Inuki, S.*; Miyagawa, T.; Oishi, S.; Ohno, H.*
J. Org. Chem. 2020, 85, 8271–8278.
doi: org/10.1021/acs.joc.0c00910

44.
Total Synthesis of Dictyodendrins A–F by the Gold-Catalyzed Cascade Cyclization of Conjugated Diyne with Pyrrole
Matsuoka, J.; Inuki, S.; Matsuda, Y.; Miyamoto, Y.; Otani, M.; Oka, M.; Oishi, S.; Ohno, H.*
Chem. Eur. J. 2020, 26, 11150–11157.

43.
Design and Discovery of Covalent α-GalCer Derivatives as Potent CD1d Ligands
Kishi, J.; Inuki, S.*; Kashiwabara, E.; Suzuki, T.; Dohmae, N.; Fujimoto, Y.*
ACS Chem. Biol. 2020, 15, 353–359.
doi: org/10.1021/acschembio.9b00700

42.
Gold(I)-Catalyzed Cascade Cyclization of Anilines with Diynes: Controllable Formation of Eight-Membered Ring-Fused Indoles and Propellane-Type Indolines
Yamaguchi, A.; Inuki, S.*; Tokimizu, Y.; Oishi, S.; Ohno, H.*
J. Org. Chem. 2020, 85, 2543–2559.
doi: org/10.1021/acs.joc.9b03256

41.
Novel Development of an Anti-Flavivirus Drug Targeting the Nucleolar Distribution of the Core Protein
Tokunaga, M.; Miyamoto, Y.; Suzuki, T.; Otani, M.; Inuki, S.; Esaki, T.; Nagao, C.; Mizuguchi, K.; Ohno, H.; Yoneda, Y.; Okamoto, T.*; Oka, M.*; Matsuura, Y.
Virology 2020, 541, 41–51.

40.
Synthetic Studies on FNC-RED and Its Analogues Containing an All syn-Cyclopentanetetrol Moiety
Inuki, S.; Sato, K.; Zui, N.; Yamaguchi, R.; Matsumaru, T.; Fujimoto, Y.*
J. Org. Chem. 2019, 84, 12680–12685.
doi: org/10.1021/acs.joc.9b02101

39.
Construction of Quaternary Carbon Stereocenter of α-Tertiary Amine through Remote C–H Functionalization of Tris Derivatives: Enantioselective Total Synthesis of Myriocin
Miyagawa, T.; Inuki, S.*; Oishi, S.; Ohno, H.*
Org. Lett. 2019, 21, 5485–5490.
doi: org/10.1021/acs.orglett.9b01778

38.
Construction of the Pyrrolo[2,3-d]carbazole Core of Spiroindoline Alkaloids by Gold-Catalyzed Cascade Cyclization of Ynamide
Matsuoka, J.; Kumagai, H.; Inuki, S.; Oishi, S.; Ohno, H.*
J. Org. Chem. 2019, 84, 9358–9363.

37.
Gold(I)-Catalyzed Cascade Cyclization Reactions of Allenynes for the Synthesis of Fused Cyclopropanes and Acenaphthenes
Ikeuchi, T.; Inuki, S.; Oishi, S.; Ohno, H.*
Angew. Chem., Int. Ed. 2019, 58, 7792–7796.

36.
Scaffold Hopping of Fused Piperidine-Type NK3 Receptor Antagonists to Reduce Environmental Impact
Yamamoto, K.; Inuki, S.; Ohno, H.; Oishi, S.*
Bioorg. Med. Chem. 2019, 27, 2019–2026.

35.
Structure-Activity Relationship Studies of Bz Amide-Containing a-GalCer Derivatives as Natural Killer T Cell Modulators
Kishi?, J.; Inuki?, S.; Hirata?, N.; Kashiwabara?, E.; Yoshidome?, D.; Ichihara?, O.; Fujimoto, Y.*
Bioorg. Med. Chem. Lett. 2019, 29, 970–973.
doi: org/10.1016/j.bmcl.2019.02.018

34.
Synthesis of Triazolo- and Oxadiazolopiperazines by Gold(I)-Catalyzed Domino Cyclization: Application to the Design of a Mitogen Activated Protein (MAP) Kinase Inhibitor
Yamamoto, K.; Yoshikawa, Y.; Ohue, M.; Inuki, S.; Ohno, H.*; Oishi, S.*
Org. Lett. 2019, 21, 373–377.

33.
Direct Synthesis of Aryl-Annulated [c]Carbazoles by Gold(I)-Catalysed Cascade Reaction of Azide-Diynes and Arenes
Kawada, Y.; Ohmura, S.; Kobayashi, M.; Nojo, W.; Kondo, M.; Matsuda, Y.; Matsuoka, J.; Inuki, S.; Oishi, S.; Wang, C.; Saito, T.; Uchiyama, M.*; Suzuki, T.*; Ohno, H.*
Chem. Sci. 2018, 9, 8416–8425.

32.
Introduction of a Polar Functional Group to the Lipid Tail of 4-epi-Jaspine B Affects Sphingosine Kinase Isoform Selectivity
Inuki, S.*; Miyagawa, T.; Oishi, S.; Ohno, H.*
Chem. Pharm. Bull. 2018, 66, 866–872.
doi: org/10.1248/cpb.c18-00366

31.
Gold(I)-Catalyzed Oxidative Cascade Cyclization of 1,4-Diyn-3-ones for the Construction of Tropone-Fused Furan Scaffolds
Hamada, N.; Yamaguchi, A.; Inuki, S.; Oishi, S.; Ohno, H.*
Org. Lett. 2018, 20, 4401–4405.

30.
Potent Th2 Cytokine-Bias of Natural Killer T Cell by CD1d Glycolipid Ligands Based on “Anchoring Effect” of Polar Groups in Their Lipid Component
Inuki, S.; Kashiwabara, E.; Hirata, N.; Kishi, J.; Nabika, E.; Fujimoto, Y.*
Angew. Chem., Int. Ed. 2018, 57, 9655–9659.
doi: org/10.1002/anie.201802983

29.
Time-lapse Monitoring of Toll-like Receptor 2 (TLR2) Ligand Internalization with Fluorescence Live-cell Imaging
Arai, Y.; Yokoyama, K.; Feng, Q.; Kawahara, Y.; Ohta, I.; Shimoyama, A.; Inuki, S.; Fukase, K.; Kabayama, K.; Fujimoto, Y.*
Org. Biomol. Chem. 2018, 16, 3824–3830.

28.
Use of a Compact Tripodal Tris(bipyridine) Ligand to Stabilize a Single-Metal-Centered Chirality: Stereoselective Coordination of Iron(II) and Ruthenium(II) on a Semirigid Hexapeptide Macrocycle
Kobayashi, Y.; Hoshino, M.; Kameda, T.; Kobayashi, K.; Akaji, K.; Inuki, S.; Ohno, H.; Oishi, S.*
Inorg. Chem. 2018, 57, 5475–5485.

27.
Site-Specific Effect of Polar Functional Group Modification in Lipids of TLR2 Ligands for Modulating the Ligand Immunostimulatory Activity
Arai, Y.; Inuki, S.; Fujimoto, Y.*
Bioorg. Med. Chem. Lett. 2018, 28, 1638–1641.

26.
Synthesis of Jaspine B Regioisomers through Palladium-Catalyzed Stereoselective Tetrahydrofuran Formation: Insight into the Ligand Recognition of Sphingosine Kinases
Miyagawa, T.; Inuki, S.; Honda, M.; Nakamura, S.; Nakanishi, I.; Fujii, N.; Oishi, S.; Ohno, H.*
Tetrahedron 2018, 74, 1802–1809.

25.
Total Synthesis and Stereochemical Revision of Stereocalpin A: Mirror-Image Approach for Stereochemical Assignments of the Peptide-Polyketide Macrocycle
Kaneda, M.; Inuki, S.; Ohno, H.; Oishi, S.*
J. Org. Chem. 2018, 83, 3047–3060.

24.
Convergent Synthesis of Digalactosyl Diacylglycerols
Inuki, S.; Kishi, J.; Kashiwabara, E.; Aiba, T.; Fujimoto, Y.*
Org. Lett. 2017, 19, 6482–6485.
doi: org/10.1021/acs.orglett.7b03043

23.
A Comprehensive Study of Interaction between Peptidoglycan Fragments and Extracelluar Domain of Mycobacterium tuberculosis Ser/Thr Kinase PknB
Wang, Q.; Marchetti, R.; Prisic, S.; Ishii, K.; Arai, Y.; Ohta, I.; Inuki, S.; Uchiyama, S.; Silipo, A.; Molinaro, A.; Husson, R. N.*; Fukase, K.; Fujimoto, Y.*
ChemBioChem 2017, 18, 2094–2098.

22.
Total Synthesis of Cardiolipins Containing Chiral Cyclopropane Fatty Acids
Inuki, S.; Ohta, I.; Ishibashi, S.; Takamatsu, M.; Fukase, K.; Fujimoto Y.*
J. Org. Chem. 2017, 82, 7832–7838.
doi: org/10.1021/acs.joc.7b00945

21.
Chemical Synthesis of D-glycero-D-manno-Heptose 1,7-Bisphosphate and Evaluation of Its Ability to Modulate NF-κB Activation
Inuki, S.; Aiba, T.; Kawakami, S.; Akiyama, T.; Inoue, J.; Fujimoto, Y.*
Org. Lett. 2017, 19, 3079–3082.
doi: org/10.1021/acs.orglett.7b01158

20.
Employing BINOL-Phosphoroselenoyl Chloride for Selective Inositol Phosphorylation and Chemical Synthesis of Glycosyl Inositol Phospholipid from Entamoeba histolytica
Aiba, T.; Suehara, S.; Choy, S.-L.; Maekawa, Y.; Lotter, H. Murai, T.; Inuki, S.; Fukase, K.; Fujimoto, Y.*
Chem. Eur. J. 2017, 23, 8304–8308.

19.
Identification of Selective Inhibitors of Sphingosine Kinases 1 and 2 through a Structure-Activity Relationship Study of 4-epi-Jaspine B
Ohno, H.*; Honda, M.; Hamada, N.; Miyagaki, J.; Iwata, A.; Otsuki, K.; Maruyama, T.; Nakamura, S.; Nakanishi, I.; Inuki, S.; Fujii, N.; Oishi, S.
Bioorg. Med. Chem. 2017, 25, 3046–3052.

18.
Formal Total Synthesis of L?Ossamine via Decarboxylative Functionalization Using Visible-Light-Mediated Photoredox Catalysis in a Flow System
Inuki, S.; Sato, K.; Fukuyama, T.; Ryu, I.; Fujimoto, Y.*
J. Org. Chem. 2017, 82, 1248–1253.
doi: org/10.1021/acs.joc.6b02531

17.
Discovery of Novel Scaffold as Indoleamine 2,3-Dioxygenase 1 (IDO1) Inhibitor Based on Pyrrolopiperazinone Alkaloid, Longamide B
Shiokawa, Z.; Kashiwabara, E.; Yoshidome, D.; Fukase, K.; Inuki, S.; Fujimoto, Y.*
ChemMedChem, 2016, 11, 2682–2689.

16.
Isolated Polar Amino Acid Residues Modulate Lipid Binding in the Large Hydrophobic Cavity of CD1d
Inuki, S.; Aiba, T.; Hirata, N.; Ichihara, O.; Yoshidome, D.; Kita, S.; Maenaka, K.; Fukase, K.; Fujimoto, Y.*
ACS Chem. Biol. 2016, 11, 3132–3139.
doi: org/10.1021/acschembio.6b00674

15.
Efficient Synthesis of (–)-Hanishin, (–)-Longamide B, and (–)-Longamide B Methyl Ester through Piperazinone Formation from 1,2-Cyclic Sulfamidates
Shiokawa, Z.; Inuki, S.; Fukase, K.; Fujimoto, Y.*
Synlett 2016, 27, 616–620.

14.
Visible-Light-Mediated Decarboxylative Benzoyloxylation of b-Hydroxy Amino Acids and Its Application to Synthesis of Functional 1,2-Amino Alcohol Derivatives
Inuki, S.; Sato, K.; Fujimoto, Y.*
Tetrahedron Lett. 2015, 56, 5787–5790.
doi: org/10.1016/j.tetlet.2015.09.012

13.
Convenient Synthesis of Spiroindole Derivatives via Palladium-Catalyzed Cyclization of Propargyl Chlorides
Iwata, A.; Inuki, S.; Oishi, S.; Fujii, N.*; Ohno. H.*
Tetrahedron 2015, 71, 6580–6585.

12.
Synthesis of Fused Tetracyclic Spiroindoles via Palladium-Catalysed Cascade Cyclisation
Iwata, A.; Inuki, S.; Oishi, S.; Fujii, N.*; Ohno. H.*
Chem.Commun. 2014, 298–300.

11.
Palladium-Catalyzed Medium-Ring Formation for Construction of the Core Structure of Laurencia Oxacycles: Synthetic Study of Laurendecumallene B
Yoshimitsu, Y.; Inuki, S.; Oishi, S.; Fujii, N.*; Ohno. H.*
Org. Lett. 2013, 15, 3046–3049.

10.
Pachastrissamine (Jaspine B) and Its Stereoisomers Inhibit Sphingosine Kinases and Atypical Protein Kinase C
Yoshimitsu, Y.; Oishi, S.; Miyagaki, J.; Inuki, S.; Ohno. H.*; Fujii, N.*
Bioorg. Med. Chem. 2011, 19, 5402–5408.

9.
Formal Total Synthesis of (+)-Lysergic Acid via Zinc(II)-Mediated Regioselective Ring-Opening Reduction of 2-Alkynyl-3-indolyloxirane
Iwata, A.; Inuki, S.; Oishi, S.; Fujii, N.*; Ohno. H.*
J. Org. Chem. 2011, 76, 5506–5512.

8.
Enantioselective Total Synthesis of (+)-Lysergic Acid, (+)-Lysergol, and (+)-Isolysergol by Palladium-Catalyzed Domino Cyclization of Allenes Bearing Amino and Bromoindolyl Groups
Inuki, S.; Iwata, A.; Oishi, S.; Fujii, N.*; Ohno. H.*
J. Org. Chem. 2011, 76, 2072–2084.

7.
Stereoselective Divergent Synthesis of Four Diastereomers of Pachastrissamine (Jaspine B)
Yoshimitsu, Y.; Inuki, S.; Oishi, S.; Fujii, N.*; Ohno. H.*
J. Org. Chem. 2010, 75, 3843–3846.

6.
Ring-Construction/Stereoselective Functionalization Cascade: Total Synthesis of Pachastrissamine (Jaspine B) through Palladium-Catalyzed Bis-cyclization of Propargyl Chlorides and Carbonates
Inuki, S.; Yoshimitsu, Y.; Oishi, S.; Fujii, N.*; Ohno. H.*
J. Org. Chem. 2010, 75, 3831–3842.

5.
Cu(II)-Mediated Oxidative Intermolecular ortho C-H Functionalisation Using Tetrahydropyrimidine as the Directing Group
Mizuhara, T.; Inuki, S.; Oishi, S.; Fujii, N.*; Ohno. H.*
Chem. Commun. 2009, 3413–3415.

4.
Ring-Construction/Stereoselective Functionalization Cascade: Total Synthesis of Pachastrissamine (Jaspine B) through Palladium-Catalyzed Bis-cyclization of Bromoallenes
Inuki, S.; Yoshimitsu, Y.; Oishi, S.; Fujii, N.*; Ohno. H.*
Org. Lett. 2009, 11, 4478–4481.

3.
Total Synthesis of (±)-Lysergic Acid, Lysergol, and Isolysergol by Palladium-Catalyzed Domino Cyclization of Amino Allenes Bearing a Bromoindolyl Group
Inuki, S.; Oishi, S.; Fujii, N.*; Ohno. H.*
Org. Lett. 2008, 10, 5239–5242.

2.
Identification of Novel Non-Peptide CXCR4 Antagonists by Ligand-Based Design Approach
Ueda, S.; Kato, M.; Inuki, S.; Ohno, H.; Evans, B.; Wang, Z.; Peiper, S. C.; Izumi, K.; Kodama, E.; Matsuoka, M.; Nagasawa, H.; Oishi, S.*; Fujii, N.*
Bioorg. Med. Chem. Lett. 2008, 18, 4124–4129.

1.
One-Pot Synthesis of Carbazoles by Palladium-Catalyzed N-Arylation and Oxidative Coupling
Watanabe, T.; Ueda, S.; Inuki, S.; Oishi, S.; Fujii, N.*; Ohno. H.*
Chem. Commun. 2007, 4516–4518.